2. Academic Validation
  3. Synthesis and applications of a novel polymer-supported EEDQ reagent

Synthesis and applications of a novel polymer-supported EEDQ reagent

  • J Comb Chem. 2007 Sep-Oct;9(5):745-7. doi: 10.1021/cc070020y.
Ramesh Kakarla 1,  Guo Li,  Samuel W Gerritz
Affiliations

Affiliation

  • 1 Early Discovery Chemistry, Bristol-Myers Squibb R&D, 5 Research Parkway, Wallingford, Connecticut 06492-7600, USA. ramesh.kakarla@bms.com
PMID: 17636942 DOI: 10.1021/cc070020y
Abstract

A simple synthetic protocol for a novel polymer-supported EEDQ reagent is reported. This reagent promotes solution-phase amide bond formation without any additives or base, as well as the selective coupling of aliphatic amines with acids in the presence of aromatic amines.

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