2. Metabolic Enzyme/Protease
  3. Endogenous Metabolite
  4. LEI-101 free base

LEI-101 free base 是一种选择性且口服生物利用度高的CB2受体激动剂，具有抑制炎症和/或氧化应激相关疾病的潜力。LEI-101 free base 对CB2受体的结合效能比CB1受体高出约100倍。其在CB2受体上的pEC50值为8，而对hERG的pKi值低于4。LEI-101可能对肾脏疾病等病症具有抑制效果。

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LEI-101 free base Chemical Structure

LEI-101 free base Chemical Structure

CAS No. : 1228660-00-1

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LEI-101 free base 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

LEI-101 free base is a selective and orally bioavailable CB2 receptor agonist with the potential to inhibit diseases associated with inflammation and/or oxidative stress. LEI-101 free base has a binding potency to CB2 receptors that is approximately 100 times higher than that to CB1 receptors. Its pEC50 value on CB2 receptors is 8, while its pKi value on hERG is less than 4. LEI-101 may have an inhibitory effect on conditions such as kidney disease[1].

分子量

472.53

Formula

C23H25FN4O4S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

LEI-101 free base 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

LEI-1011228660-00-1LEI101LEI 101Endogenous MetaboliteInhibitorinhibitorinhibit

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