2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. nAChR
  4. UB-165 fumarate

UB-165 fumarate 是 nAChR 的激动剂，是 α3β2 亚型的全激动剂，α4β2* 亚型的部分激动剂，其在大鼠脑中测得的结合到 [3H]-nicotine 的 Ki 值为 0.27 nM。

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UB-165 fumarate Chemical Structure

UB-165 fumarate Chemical Structure

CAS No. : 2454492-43-2

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Other Forms of UB-165 fumarate:

UB-165 fumarate 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

UB-165 fumarate is a nAChR agonist, being a full agonist of the α3β2 isoform and a partial agonist of the α4β2* isoform, with a Ki value of 0.27 nM for [3H]-nicotine binding in rat brain[1].

IC50 & Target

Ki: 0.27 nM (nicotine in rat brain)[1].
体外研究
(In Vitro)

UB-165 fumarate stimulates [3H]-dopamine release from striatal synaptosomes with an EC50 value of 88 nM[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

UB-165 fumarate 相关抗体:
分子量

350.80

Formula

C17H19ClN2O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

UB-165 fumarate 相关分类

  • 摩尔计算器

  • 稀释计算器

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

UB-1652454492-43-2UB165UB 165nAChRNicotinic acetylcholine receptorsInhibitorinhibitorinhibit

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产品名称：
UB-165 fumarate
目录号：
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