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  4. YM-44781 free acid

YM-44781 free acid是一种非肽类的神经肽受体拮抗剂，具有高效的NK(2)和NK(1)受体拮抗活性。YM-44781在NK(2)受体上表现出显著的结合亲和力(pKi = 9.94)，并且在NK(1)受体上也有较高的结合亲和力(pKi = 9.09)。此外，YM-44781在选择性NK(1)受体激动剂诱导的膀胱收缩中也显示出了显著的抑制作用。

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YM-44781 free acid Chemical Structure

YM-44781 free acid Chemical Structure

CAS No. : 173943-29-8

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YM-44781 free acid 相关抗体

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生物活性

YM-44781 free acid is a non-peptide neuropeptide receptor antagonist with efficient NK(2) and NK(1) receptor antagonist activity. YM-44781 exhibits significant binding affinity on the NK(2) receptor (pKi = 9.94) and also on the NK(1) receptor Higher binding affinity (pKi = 9.09). In addition, YM-44781 also showed significant inhibitory effects on bladder contraction induced by selective NK(1) receptor agonists[1].

分子量

568.51

Formula

C31H32Cl2FN3O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

YM-44781 free acid 相关分类

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  • Do most proteins show cross-species activity?

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Keywords:

YM-44781173943-29-8YM44781YM 44781OthersInhibitorinhibitorinhibit

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