1. Metabolic Enzyme/Protease
  2. Endogenous Metabolite
  3. AKR1C2/3-IN-2

AKR1C2/3-IN-2是一种潜在的AKR1C3抑制剂,具有选择性抑制AKR1C3的活性。AKR1C2/3-IN-2能够阻止AKR1C3介导的睾酮(T)生成和PSA诱导,影响前列腺癌细胞的内分泌活动。AKR1C2/3-IN-2显示出对其他AKR1C酶的选择性,表明其在抑制耐药性前列腺癌中的潜在应用。AKR1C2/3-IN-2与COX异构酶无抑制活性,进一步强调了其作为前列腺癌抑制化合物的特异性。

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AKR1C2/3-IN-2 Chemical Structure

AKR1C2/3-IN-2 Chemical Structure

CAS No. : 56600-73-8

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  • 生物活性

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生物活性

AKR1C2/3-IN-2 is a potential AKR1C3 inhibitor with selective AKR1C3 activity. AKR1C2/3-IN-2 is able to block AKR1C3-mediated testosterone (T) production and PSA induction, affecting the endocrine activity of prostate cancer cells. AKR1C2/3-IN-2 shows selectivity over other AKR1C enzymes, indicating its potential application in inhibiting drug-resistant prostate cancer. AKR1C2/3-IN-2 has no inhibitory activity against COX isomerases, further emphasizing its specificity as a prostate cancer inhibitory compound[1].

分子量

244.29

Formula

C15H16O3

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

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产品名称:
AKR1C2/3-IN-2
目录号:
HY-121656
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