2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. CB2R agonist 1

CB2R agonist 1 是一种大麻素受体亚型 2 (CB2R) 的选择性配体，EC50 值为 0.56 µM。CB2R agonist 1 对人 CB2R 和 CB1R 分别具有高亲和力及优异选择性。CB2R agonist 1 调节促炎细胞因子和抗炎细胞因子的产生，发挥免疫调节作用。

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CB2R agonist 1 Chemical Structure

CB2R agonist 1 Chemical Structure

CAS No. : 1817633-49-0

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CB2R agonist 1 相关抗体

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CB1 CB2

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CB2R agonist 1 is a selective ligand of cannabinoid receptor subtype 2 (CB2R) with an EC50 value of 0.56 µM. CB2R agonist 1 has high affinity and excellent selectivity for human CB2R and CB1R respectively. CB2R agonist 1 regulates the production of pro-inflammatory cytokines and anti-inflammatory cytokines and play an immunomodulatory role[1].

IC50 & Target[1]

CB2R

0.56 μM (EC50)

体外研究
(In Vitro)

CB2R agonist 1 (Compound 4) (1 μM 和 10 μM；24 h) 以浓度依赖性方式增加单核细胞和巨噬细胞中 IL-4、IL-10 抗炎细胞因子的产生，减少 TNF-α、IFN-γ、IL-1β、IL-6 促炎性细胞因子的产生[1]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

CB2R agonist 1 相关抗体:
分子量

340.50

Formula

C22H32N2O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CB2R agonist 1 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CB2R agonist 11817633-49-0Cannabinoid ReceptorMonocytesMacrophagesTNF-αIFN-γIL-1βIL-6IL-4IL-10Inhibitorinhibitorinhibit

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