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Droxicam (Ombolan) 是一种非甾体类抗炎剂,具有很强的镇痛作用。Droxicam 通过抑制 PGE2 发挥作用,其特点是 Piroxicam (HY-B0253) 的前体药物。Droxicam 具有良好的耐受性,在所述粘膜中有轻微的副作用。Droxicam 不会对猫的心血管或呼吸系统产生影响,但会抑制小鼠的腹膜毛细血管通透性。

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Droxicam Chemical Structure

Droxicam Chemical Structure

CAS No. : 90101-16-9

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Droxicam (Ombolan) is a non-steroidal anti-inflammatory agent, with strong analgesic activity. Droxicam acts by inhibiting PGE2 varies, and is characterised by being a pro-drug of Piroxicam (HY-B0253). Droxicam is well tolerated with slight side effects in the said mucosa. Droxicam does not show cardiovascular or respiratory effects in cats, and inhibits peritoneal capillary permeability in mouse[1][2].

体内研究
(In Vivo)

Droxicam (0.25 和 0.5 mg/kg;口服) 在角叉菜胶诱导的大鼠水肿中表现出高抗炎活性[1]
Droxicam (ED50, p.o.; 5, 6, 7, 8 h; 7.5, 12.9, 4.8, 8.4 mg/kg) 在大鼠中对制霉菌素诱导的水肿表现出高抗炎活性[1]
Droxicam (ED50,口服,1、2、3、4 小时:0.51、0.94、1.56、4.88 mg/kg) 对紫外线光诱导红斑的豚鼠,显示出保护作用[1]
Droxicam (0.1 mg/kg, 0.33 mg/kg, 1 mg/kg; po; 每日一次) 在注射 Mycobacterium butyricum 的大鼠中显示出良好的抗关节炎活性,可抵抗原发性和继发性病变[1]
Droxicam 在防止小鼠扭体方面表现出很强的镇痛活性,对由苯基苯醌诱导、乙酰胆碱溴化物诱导的小鼠,ED50 分别为 5.3 mg/kg 和 1.1 mg/kg[1]
Droxicam (ED50=0.081 mg/kg; po) 保护大鼠免受蓖麻油引起的腹泻[1]
Droxicam 显著抑制小鼠腹膜毛细血管通透性[1]
Droxicam 在 Irwin 试验中,不会改变大鼠的行为 (80 mg/kg,i.p.) 和小鼠的行为 (160 mg/kg,p.o.)[1]
Droxicam 在大鼠中不表现出排尿酸活性,在麻醉猫中既不表现出心血管或呼吸作用,也不改变它们对乙酰胆碱、去甲肾上腺素和组胺给药的反应[1]

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

357.34

Formula

C16H11N3O5S

CAS 号
中文名称

屈昔康

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献

Droxicam 相关分类

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  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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