2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. Enadoline

Enadoline  (Synonyms: 依那朵林; CI-977)

目录号: HY-105235
产品使用指南

摩尔计算器

Enadoline (CI-977) 是一种高选择性、能透过血脑屏障的、非肽 κ 阿片受体 (KOR) 激动剂 (Ki=1.25 nM)。具有抗伤害作用。

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Enadoline Chemical Structure

Enadoline Chemical Structure

CAS No. : 124378-77-4

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Customer Review

Enadoline 相关抗体

Top Publications Citing Use of Products

查看 Opioid Receptor 亚型特异性产品:

查看所有亚型
μ Opioid Receptor/MOR κ Opioid Receptor/KOR δ Opioid Receptor/DOR NOP Receptor/ORL1

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Enadoline (CI-977) is a highly selective, brain-penetrating, and nonpeptide kappa-opioid receptor (KOR) agonist (Ki=1.25 nM). Antinociceptive effects[1][2].

体内研究
(In Vivo)

Enadoline (i.v.; dose of e 15 min before surgery; male Sprague-Dawley rats) dose-dependently (1-100 μg/kg) blocks the development of thermal hyperalgesia as well as static and dynamic allodynia for over 24 h with respective MEDs (minimum effective doses) of < or = 1, 10 and 10 μg/kg[2].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

396.52

Formula

C24H32N2O3
CAS 号
中文名称

依那朵林
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Enadoline 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Enadoline124378-77-4CI-977依那朵林CI977CI 977Opioid ReceptorselectivebrainpenetratingnonpeptideantinociceptiveInhibitorinhibitorinhibit

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