2. Protein Tyrosine Kinase/RTK
  3. Ephrin Receptor
  4. EphA2 agonist 2

EphA2 agonist 2 (Lead compound) 是一种选择性的 EphA2 激动剂，具有抗肿瘤活性。EphA2 agonist 2 能透过血脑屏障

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EphA2 agonist 2 Chemical Structure

EphA2 agonist 2 Chemical Structure

CAS No. : 2169273-66-7

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EphA2 agonist 2 相关抗体

Top Publications Citing Use of Products

查看 Ephrin Receptor 亚型特异性产品:

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EphA2 EphA3 EphA4

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

EphA2 agonist 2 (Lead compound) is a selective EphA2 agonist with antitumor activities. EphA2 agonist 2 can cross the BBB[1].

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
U-251 IC50
2.1 μM
Compound: Table 4, Lead cpd
Antiproliferative activity against human U251 cells overexpressing EPHA2 assessed as reduction in cell viability incubated for 48 hrs by MTT assay
Antiproliferative activity against human U251 cells overexpressing EPHA2 assessed as reduction in cell viability incubated for 48 hrs by MTT assay
[PMID: 32828423]
U-251 IC50
5.2 μM
Compound: Table 4, Lead cpd
Antiproliferative activity against wild-type human U251 cells assessed as reduction in cell viability incubated for 48 hrs by MTT assay
Antiproliferative activity against wild-type human U251 cells assessed as reduction in cell viability incubated for 48 hrs by MTT assay
[PMID: 32828423]
体外研究
(In Vitro)

EphA2 agonist 2 (Lead compound) shows antiproliferation activity with IC50 values of 2.1 ± 1.05 μM and 5.2 ± 2.56 μM against U251 EphA2 overexpressed and U251 wild type cells, respectively[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

EphA2 agonist 2 相关抗体:
分子量

772.94

Formula

C40H56N10O6
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

EphA2 agonist 2 相关分类

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

EphA2 agonist 22169273-66-7Ephrin ReceptorU251antitumorBBBInhibitorinhibitorinhibit

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产品名称：
EphA2 agonist 2
目录号：
HY-146141
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