2. GPCR/G Protein Neuronal Signaling
  3. Melanocortin Receptor
  4. GPS1573

GPS1573 是一种黑素皮质素 2 型受体 (MC2R) 的非竞争性拮抗剂，剂量依赖性地拮抗 ACTH 刺激的 MC2R 活性 (IC50=66 nM)。GPS1573 因其对 MC2R 的高选择性拮抗作用，可用于库欣病的研究。

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Custom Peptide Synthesis

GPS1573 Chemical Structure

GPS1573 Chemical Structure

CAS No. : 2445822-54-6

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GPS1573 相关抗体

Top Publications Citing Use of Products

查看 Melanocortin Receptor 亚型特异性产品:

查看所有亚型
MC1R MC3R MC2R MC4R MC5R

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GPS1573 is a noncompetitive antagonist of melanocortin type 2 receptor (MC2R) that dose-dependently antagonizes ACTH-stimulated MC2R activity (IC50=66 nM). GPS1573 can be used in the study of Cushing's disease due to its highly selective antagonism of MC2R[1].

分子量

1788.20

Formula

C86H138N28O14
CAS 号
Sequence

{Nle}-Pro-{d-Phe}-Arg-{d-Trp}-Phe-Lys-Ala-Val-Gly-Lys-Lys-Arg-Arg-NH2
Sequence Shortening

{Nle}-P-{d-Phe}-R-{d-Trp}-FKAVGKKRR-NH2
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GPS1573 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPS15732445822-54-6GPS 1573GPS-1573Melanocortin ReceptorMC ReceptorAntagonistnon-competitivehighly selectiveCushing diseaseMC2RInhibitorinhibitorinhibit

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产品名称：
GPS1573
目录号：
HY-P10571
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