2. GPCR/G Protein
  3. GnRH Receptor
  4. Histrelin

Histrelin  (Synonyms: 组氨瑞林)

目录号: HY-P0056
产品使用指南

摩尔计算器

Histrelin，一种 GnRH 类似物，是一种 GnRH 受体激动剂。Histrelin 可增加血清中促黄体激素(LH)、促卵泡激素 (FSH) 和睾酮水平。Histrelin 可用于前列腺癌、子宫内膜异位症的研究。

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Custom Peptide Synthesis

Histrelin Chemical Structure

Histrelin Chemical Structure

CAS No. : 76712-82-8

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Histrelin 的其他形式现货产品:

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Other Forms of Histrelin:

Histrelin 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Histrelin, a GnRH analogue, is a GnRH Receptor agonist. Histrelin increases serum luteinising hormone (LH), follicle stimulating hormone (FSH) and testosterone levels. Histrelin can be used in the research of prostate cancer, endometriosis[1][2][5].

IC50 & Target

GnRH Receptor[1]
体外研究
(In Vitro)

Histrelin (10-100 nM) stimulates the release of vasopressin (VP) from from isolated rat hypothalamo-neurohypophysial explants[4].
Histrelin (100 nM) stimulates oxytocin (OT) release from the rat hypothalamo-neurohypophysial system[5].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Histrelin 相关抗体:
体内研究
(In Vivo)

Histrelin (0.1 mg/kg，皮下注射) 可恢复 Csfmop/Csfmop 小鼠[2]中的循环 LH 浓度。
Histrelin （10,30 或 100 μg/天，皮下注射)会减少兔子的子宫内膜腺体数量并使间质萎缩[3]。

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Csfmop/Csfmop mice [2]
Dosage: 0.001, 0.05, and 0.1 mg/kg
Administration: Subcutaneous injection
Result: Increased serum FSH concentrations by 4-fold.
Animal Model: Rabbits[3]
Dosage: 10, 30, or 100 μg /day
Administration: Subcutaneous injection for 4 weeks
Result: Caused a regression of the endometrial glands and a thinning of the stroma.
Clinical Trial
分子量

1323.50

Formula

C66H86N18O12
CAS 号
Sequence

{Pyr}-His-Trp-Ser-Tyr-D-His(Bzl)-Leu-Arg-Pro-NHEt
Sequence Shortening

{Pyr}-HWSYHLRP-NHEt
中文名称

组氨瑞林
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Histrelin 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Histrelin76712-82-8组氨瑞林GnRH ReceptorGonadotropin releasing hormone receptorGNRHRProstate cancerendometriosisLHvasopressinVPFSHH-N systermInhibitorinhibitorinhibit

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