2. Anti-infection Metabolic Enzyme/Protease
  3. HIV Protease
  4. HIV-1 protease-IN-7

HIV-1 protease-IN-7 (化合物 16) 是一种口服有效的 HIV-1 蛋白酶抑制剂 (IC50=3.52 nM, EC50=37 nM)。

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Custom Peptide Synthesis

HIV-1 protease-IN-7 Chemical Structure

HIV-1 protease-IN-7 Chemical Structure

CAS No. : 2916441-36-4

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HIV-1 protease-IN-7 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

HIV-1 protease-IN-7 (compound 16) is an orally active HIV-1 protease inhibitor (IC50=3.52 nM, EC50=37 nM)[1].

IC50 & Target

HIV-1 protease[1].
体内研究
(In Vivo)

HIV-1 protease-IN-7 (2.57 mg/kg; p.o.; single) exhibits good plasma total clearance and oral bioavailability[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male Sprague-Dawley rats (8-week-old)[1].
Dosage: 2.57 mg/kg (2 μM/kg)
Administration: Oral administration; single.
Result: 1.19 Pharmacokinetic Parameters of HIV-1 protease-IN-7 in male Sprague-Dawley rats[1].
metabolic stability rat/human (%) CLtot (mL/min/kg) Vdss (L/kg) t1/2 (h) F (%) serum fu(%)
PO (2.57 mg/kg) 63/23 8.2 1.9 3.9 3.3 0.1
分子量

1285.68

Formula

C68H104N10O12S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

HIV-1 protease-IN-7 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

HIV-1 protease-IN-72916441-36-4HIV ProteaseHIV-1Inhibitorinhibitorinhibit

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产品名称：
HIV-1 protease-IN-7
目录号：
HY-151250
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