1. GPCR/G Protein
  2. Bombesin Receptor
  3. ICI 216140

ICI 216140 是一种 GRP/蛙皮素受体 2 (GRP/bombesin receptor 2) 拮抗剂,其 IC50 值为 2 nM。ICI 216140 可以减少 Bombesin (HY-P0195) 刺激的胰淀粉酶分泌,并减轻 Bombesin (HY-P0195) 刺激的血压升高。

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Custom Peptide Synthesis

ICI 216140 Chemical Structure

ICI 216140 Chemical Structure

CAS No. : 124001-41-8

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

ICI 216140 is a GRP/bombesin receptor 2 antagonist with the IC50 of 2 nM. ICI 216140 can reduce Bombesin (HY-P0195)-stimulated pancreatic amylase secretion and attenuates Bombesin (HY-P0195)-stimulated increases in blood pressure[1][2].

分子量

916.08

Formula

C45H65N13O8

CAS 号
Sequence

{N-Isobutyryl}-His-Trp-Ala-Val-{d-(Ala)}-His-Leu-NHMe

Sequence Shortening

{N-Isobutyryl}-HWAV-{d-(Ala)}-HL-NHMe

运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Inquiry Information

产品名称:
ICI 216140
目录号:
HY-P3112
需求量: