2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. LY2048978

LY2048978 是一种非选择性的阿片受体 (Opioid Receptor) 拮抗剂，在体外对人 mu，kappa 和 delta 阿片受体的 Ki分别为 0.287, 0.471 和 1.05 nM。LY2048978 可用于重度抑郁症和酒精使用障碍的研究。

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LY2048978 Chemical Structure

LY2048978 Chemical Structure

CAS No. : 676495-11-7

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LY2048978 相关抗体

Top Publications Citing Use of Products

查看 Opioid Receptor 亚型特异性产品:

查看所有亚型
μ Opioid Receptor/MOR κ Opioid Receptor/KOR δ Opioid Receptor/DOR NOP Receptor/ORL1

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

LY2048978 is a non-selective opioid receptor antagonist with Ki of 0.287, 0.471 and 1.05 nM for human mu, kappa and delta opioid receptors in vitro, respectively. LY2048978 can be used in the research of major depressive disorder and alcohol use disorder[1].

IC50 & Target[1]

μ Opioid Receptor/MOR

0.287 nM (Ki)

κ Opioid Receptor/KOR

0.471 nM (Ki)

δ Opioid Receptor/DOR

1.05 nM (Ki)

分子量

312.41

Formula

C19H24N2O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

LY2048978 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

LY2048978676495-11-7LY 2048978LY-2048978Opioid Receptornonselectiveantagonistquality controlmajor depressionInhibitorinhibitorinhibit

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目录号：
HY-118615
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