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  4. 8-(3-Chlorostyryl)caffeine

8-(3-Chlorostyryl)caffeine  (Synonyms: CSC)

目录号: HY-103164A
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8-(3-Chlorostyryl)caffeine (CSC)是一种腺苷拮抗剂，具有对A2a腺苷受体的选择性活性。8-(3-Chlorostyryl)caffeine在大鼠大脑的放射配体结合实验中显示出520倍选择性。8-(3-Chlorostyryl)caffeine对腺苷酰化酶的拮抗作用在大鼠嗜铬细胞中显示出22倍的选择性8-(3-Chlorostyryl)caffeine与A1选择性拮抗剂CPX共同施用时，亦能进一步增加运动活性。8-(3-Chlorostyryl)caffeine在灵长类动物的线粒体中表现出良好的MAO-B抑制活性。8-(3-Chlorostyryl)caffeine的A2A受体亲和力也表现优异。

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8-(3-Chlorostyryl)caffeine Chemical Structure

8-(3-Chlorostyryl)caffeine Chemical Structure

CAS No. : 148589-13-3

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Other Forms of 8-(3-Chlorostyryl)caffeine:

8-(3-Chlorostyryl)caffeine 相关抗体

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生物活性

8-(3-Chlorostyryl)caffeine (CSC) is an adenosine antagonist with selective activity at the A2a adenosine receptor. 8-(3-Chlorostyryl)caffeine showed 520-fold selectivity in radioligand binding experiments in rat brain. Antagonism of adenylylase by 8-(3-Chlorostyryl)caffeine shows 22-fold selectivity in rat chromaffin cells When 8-(3-Chlorostyryl)caffeine is co-administered with the A1-selective antagonist CPX, It can also further increase exercise activity. 8-(3-Chlorostyryl)caffeine exhibits good MAO-B inhibitory activity in primate mitochondria. 8-(3-Chlorostyryl)caffeine also has excellent A2A receptor affinity[1].

分子量

330.77

Formula

C16H15ClN4O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

8-(3-Chlorostyryl)caffeine 相关分类

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Keywords:

8-(3-Chlorostyryl)caffeine148589-13-3CSCOthersInhibitorinhibitorinhibit

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