2. GPCR/G Protein
  3. GPR4
  4. GPR4 antagonist 1

GPR4 antagonist 1 是 GPR4 的拮抗剂，其 IC50 值为 189 nM。

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GPR4 antagonist 1 Chemical Structure

GPR4 antagonist 1 Chemical Structure

CAS No. : 1197879-16-5

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1 mg ￥2320
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5 mg ￥5800
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GPR4 antagonist 1 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GPR4 antagonist 1 is a GPR4 antagonist, with an IC50 of 189 nM.

IC50 & Target

IC50: 189 nM (GPR4)[1].
细胞效力
(Cellular Effect)
Cell Line Type Value Description References
HeLa IC50
0.11 μM
Compound: 39c
Antagonist activity at human GPR4 expressed in human HeLa cells assessed as inhibition of pH-induced cAMP accumulation preincubated for 15 mins followed by cAMP addition measured after 60 mins by HTRF method
Antagonist activity at human GPR4 expressed in human HeLa cells assessed as inhibition of pH-induced cAMP accumulation preincubated for 15 mins followed by cAMP addition measured after 60 mins by HTRF method
[PMID: 28689977]
分子量

431.62

Formula

C27H37N5
CAS 号
性状

油状物

颜色

Light yellow to yellow

运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Pure form -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
纯度 & 产品资料

纯度: 98.92%

COA (262 KB) HNMR (269 KB) LCMS (267 KB)

产品使用指南 (1538 KB)
参考文献

GPR4 antagonist 1 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GPR4 antagonist 11197879-16-5GPR4G Protein-Coupled Receptor 4Inhibitorinhibitorinhibit

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产品名称：
GPR4 antagonist 1
目录号：
HY-101536
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