PKD Inhibitors

PKD1, IC₅₀: 1 nM

PKD2, IC₅₀: 2.5 nM

PKD3, IC₅₀: 2 nM

PKD1, IC₅₀: 182 nM

PKD2, IC₅₀: 280 nM

PKD3, IC₅₀: 227 nM

PKD1, IC₅₀: 154.6 nM

PKD2, IC₅₀: 133.4 nM

PKD3, IC₅₀: 109.4 nM

PKD1, IC₅₀: 28.3 nM

PKD2, IC₅₀: 58.7 nM

PKD3, IC₅₀: 53.2 nM

PKD1, IC₅₀: 1 nM

PKD2, IC₅₀: 2.5 nM

PKD3, IC₅₀: 2 nM

PKD1, IC₅₀: 3.2 μM

Cellular PKD2, IC₅₀: 0.6 μM

Cellular PKD3, IC₅₀: 0.7 μM

PKD1, IC₅₀: 1 nM

PKD2, IC₅₀: 2.5 nM

PKD3, IC₅₀: 2 nM

PKD1, IC₅₀: 1 nM

PKD2, IC₅₀: 9 nM

PKD3, IC₅₀: 1 nM

PKD1, IC₅₀: 108 nM

Cellular PKD2, IC₅₀: 94 nM

PKD3, IC₅₀: 108 nM

PKD1, IC₅₀: 0.6 nM

PKD1, IC₅₀: 35 ± 10 nM

PKD2, IC₅₀: 35 ± 5 nM

PKD3, IC₅₀: 17 ± 8 nM