2. GPCR/G Protein
  3. Adenosine Receptor
  4. Adenosine receptor antagonist 5

Adenosine receptor antagonist 5 

目录号: HY-162787
产品使用指南

摩尔计算器

Adenosine receptor antagonist 5 (Compound 39) 是人类腺苷 A3 受体 (hA3R) 的选择性拮抗剂，Ki 为 12 nM。Adenosine receptor antagonist 5 可在 NCI-H1792 细胞中抑制 IB-MECA (HY-13591) 诱导的 cAMP 的积累，抑制癌细胞 LK-2 和 NCI-H1792 的增殖。Adenosine receptor antagonist 5 在人肝微粒体中表现出快速的代谢率。

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Adenosine receptor antagonist 5 Chemical Structure

Adenosine receptor antagonist 5 Chemical Structure

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Adenosine receptor antagonist 5 相关抗体

Top Publications Citing Use of Products

查看 Adenosine Receptor 亚型特异性产品:

查看所有亚型
Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Adenosine receptor antagonist 5 (Compound 39) is a selective antagonist for human adenosine A3 receptor (hA3R) with Ki of 12 nM. Adenosine receptor antagonist 5 inhibits IB-MECA (HY-13591)-induced cAMP accumulation in NCI-H1792 cell, inhibits the proliferation of cancer cell LK-2 and NCI-H1792. Adenosine receptor antagonist 5 exhibits a fast metabolic rate in human liver microsomes[1].

IC50 & Target

human A3

12 nM (Ki)

分子量

470.10

Formula

C17H11BrCl2N4O3
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Adenosine receptor antagonist 5 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Adenosine receptor antagonist 5Adenosine receptor antagonist5Adenosine receptor antagonist-5Adenosine ReceptorP1 receptorLK-2NCI-H1792selectiveInhibitorinhibitorinhibit

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Adenosine receptor antagonist 5
目录号：
HY-162787
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