2. GPCR/G Protein Neuronal Signaling
  3. Cannabinoid Receptor
  4. CB2 receptor antagonist 1

己基间苯二酚衍生物29被证明是一种CB2选择性竞争性拮抗剂/反向激动剂，具有良好的效力。橄榄醇和5-（2-甲基辛烷-2-基）间苯二酚衍生物23和24均表现出显着的抗伤害感受活性，化合物24被证明能够激活大麻素和TRPV1受体。

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CB2 receptor antagonist 1 Chemical Structure

CB2 receptor antagonist 1 Chemical Structure

CAS No. : 2772693-05-5

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CB2 receptor antagonist 1 相关抗体

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CB1 CB2

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Hexyl resorcinol derivative 29 has been proved to be a CB2 selective competitive antagonist / reverse agonist with good potency. Olivanol and 5- (2-methyloctane-2-yl) resorcinol derivatives 23 and 24 showed significant antinociceptive activity. Compound 24 was shown to activate cannabinoid and TRPV1 receptors.

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
CHO EC50
173.6 nM
Compound: 29
Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liquid scintillation counting assay
Agonist activity at human CB2 receptor expressed in CHO cell membrane assessed as inhibition of [35S]-GTPgammaS binding incubated for 1 hr by by liquid scintillation counting assay
[PMID: 32340793]
分子量

445.68

Formula

C28H47NO3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CB2 receptor antagonist 1 相关分类

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Keywords:

CB2 receptor antagonist 12772693-05-5Cannabinoid ReceptorInhibitorinhibitorinhibit

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