2. Metabolic Enzyme/Protease Neuronal Signaling GPCR/G Protein
  3. FAAH Cannabinoid Receptor
  4. CB2R/FAAH modulator-2

CB2R/FAAH modulator-2 (compound 26) 是一种双重靶向调节剂，可以作为 CB2R 激动剂和 FAAH 抑制剂。CB2R/FAAH modulator-2 作用于 CB2R 和 CB1R 的 Ki 值分别是 10.8 和 152.9 nM，作用于FAAH 的 IC50 值为 6.2 μM。CB2R/FAAH modulator-2 可用于癌症、神经退行性疾病中发生的有害炎症级联反应以及 COVID-19 感染相关研究。

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CB2R/FAAH modulator-2 Chemical Structure

CB2R/FAAH modulator-2 Chemical Structure

CAS No. : 2876918-68-0

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规格 价格 是否有货
5 mg ￥900
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10 mg ￥1500
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CB2R/FAAH modulator-2 相关抗体

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CB1 CB2

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CB2R/FAAH modulator-2 (compound 26) is a dual targeting modulator that acts as a CB2R agonist and FAAH inhibitor. The Ki values for CB2R/FAAH modulator-2 are 10.8 and 152.9 nM for CB2R and CB1R, respectively, and the IC50 value for FAAH is 6.2 μM. CB2R/FAAH modulator-2 can be used in studies related to cancer, deleterious inflammatory cascades occurring in neurodegenerative diseases, and COVID-19 infection[1].

IC50 & Target[1]

CB1

152.9 nM (Ki)

CB2

10.8 nM (Ki)

体外研究
(In Vitro)

CB2R/FAAH modulator-2 (compound 26)(10 μM) reduces the production of the pro-inflammatory cytokines TNFα, IFN-γ, IL-1β and IL6 in unstimulated monocytes and macrophages[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

CB2R/FAAH modulator-2 相关抗体:
分子量

367.52

Formula

C24H33NO2
CAS 号
性状

固体

颜色

Light yellow to yellow

运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
纯度 & 产品资料
参考文献

CB2R/FAAH modulator-2 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CB2R/FAAH modulator-22876918-68-0FAAHCannabinoid ReceptorFatty acid amide hydrolaseCB2RCB1RcancerneurodegenerativeinflammatoryCOVID-19Inhibitorinhibitorinhibit

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