2. Cell Cycle/DNA Damage Stem Cell/Wnt
  3. Casein Kinase
  4. CK1α degrader-1

CK1α degrader-1 (Compound 82) 是一种具有口服活性的 CK1α 降解剂，DC50 为 0.105 μM。CK1α degrader-1可用于癌症的研究。

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CK1α degrader-1 Chemical Structure

CK1α degrader-1 Chemical Structure

CAS No. : 2881012-96-8

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CK1α degrader-1 相关抗体

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

CK1α degrader-1 (Compound 82) is an orally active CK1α degrader with a DC50 of 0.105 μM. CK1α degrader-1 can be used for the research of cancer[1].

体内研究
(In Vivo)


药代动力学分析[1]

Route Dose (mg/kg) CL (mL/min/kg) C0 (ng/mL) t1/2 (hr) Vss (L/kg)
i.v. 2 10.5 6796 1.34 0.85
Route Dose (mg/kg) Cmax (ng/mL) Tmax (h) T1/2 (h) AUC(0-inf) (ng·h/mL) F (%)
p.o. 10 6080 0.67 2.03 13264 85

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

466.92

Formula

C24H23ClN4O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

CK1α degrader-1 相关分类

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  • 稀释计算器

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Keywords:

CK1α degrader-12881012-96-8Casein KinaseCK1αcancerorally activeInhibitorinhibitorinhibit

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目录号：
HY-160532
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