1. Metabolic Enzyme/Protease
  2. Cytochrome P450
  3. CYP1B1 ligand 3

CYP1B1 ligand 3 (Compound A1) 是细胞色素 P450 酶 CYP1B1 的选择性抑制剂,IC50 为 11.9 nM。CYP1B1 ligand 3 可用于合成 PROTAC CYP1B1 degrader-2 (HY-158429)。

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CYP1B1 ligand 3 Chemical Structure

CYP1B1 ligand 3 Chemical Structure

CAS No. : 65823-65-6

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  • 生物活性

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生物活性

CYP1B1 ligand 3 (Compound A1) is a selective inhibitor for cytochrome P450 enzyme CYP1B1 with an IC50 of 11.9 nM. CYP1B1 ligand 3 can be utilized for the synthesis of PROTAC CYP1B1 degrader-2 (HY-158429)[1].

IC50 & Target

CYP1B1

11.9 nM (IC50)

CYP1A1

278.7 nM (IC50)

CYP1A2

3913.5 nM (IC50)

分子量

369.89

Formula

C18H12ClN3S2

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
CYP1B1 ligand 3
目录号:
HY-159006
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