2. Neuronal Signaling GPCR/G Protein
  3. Serotonin Transporter 5-HT Receptor
  4. DSP-1053 benzenesulfonate

DSP-1053 是一种苄基哌啶衍生物，一种有效的血清素转运蛋白 (SERT) 抑制剂，Ki 值为 1.02 nM。DSP-1053 显示 5-HT1A 受体部分激动活性，Ki 值为 5.05 nM。DSP-1053 具有抗抑郁活性。

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DSP-1053 benzenesulfonate Chemical Structure

DSP-1053 benzenesulfonate Chemical Structure

CAS No. : 1176326-78-5

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DSP-1053 benzenesulfonate 的其他形式现货产品:

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Other Forms of DSP-1053 benzenesulfonate:

DSP-1053 benzenesulfonate 相关抗体

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5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

DSP-1053, a benzylpiperidine derivative, is a potent serotonin transporter (SERT) inhibitor with a Ki of 1.02 nM. DSP-1053 shows partial 5-HT1A receptor agonistic activity with a Ki of 5.05 nM. DSP-1053 has antidepressant activity[1].

IC50 & Target[1]

5-HT1A Receptor

5.05 nM (Ki)

Clinical Trial
分子量

660.62

Formula

C32H38BrNO7S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

DSP-1053 benzenesulfonate 相关分类

  • 摩尔计算器

  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

DSP-10531176326-78-5DSP1053DSP 1053Serotonin Transporter5-HT Receptor5-HTTSERTSLC6A4Serotonin Receptor5-hydroxytryptamine ReceptorBenzylpiperidine,?Serotonin Transporter5-HT1AantidepressantInhibitorinhibitorinhibit

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