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  4. EST64454 maleate

EST64454 maleate 是一种高溶解度的 σ1 受体拮抗剂，具有强效的镇痛特性，可用于疼痛抑制。EST64454 maleate 在各种物种中均表现出极佳的代谢稳定性，在啮齿动物中具有良好的药代动力学特征。EST64454 maleate 因其在 Caco-2 细胞中具有良好的水溶性和高渗透性而被认定为有前途的临床候选化合物。

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EST64454 maleate Chemical Structure

EST64454 maleate Chemical Structure

CAS No. : 2088272-67-5

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EST64454 maleate 相关抗体

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生物活性

EST64454 maleate is a highly soluble σ1 receptor antagonist, demonstrating potent antinociceptive properties for pain treatment. EST64454 maleate exhibits excellent metabolic stability across various species and possesses an adequate pharmacokinetic profile in rodents. EST64454 maleate has been identified as a promising clinical candidate due to its favorable aqueous solubility and high permeability in Caco-2 cells.

分子量

480.46

Formula

C22H26F2N4O6
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

EST64454 maleate 相关分类

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  • Do most proteins show cross-species activity?

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Keywords:

EST644542088272-67-5EST 64454EST-64454OthersInhibitorinhibitorinhibit

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EST64454 maleate
目录号：
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