2. Apoptosis Epigenetics
  3. Apoptosis Epigenetic Reader Domain
  4. GSK778 hydrochloride

GSK778 hydrochloride  (Synonyms: iBET-BD1 hydrochloride)

目录号: HY-136570A
产品使用指南

摩尔计算器

GSK778 (iBET-BD1) hydrochloride 是一种有效和选择性的 BET 蛋白 BD1 溴结构域的抑制剂，IC50 值为 75 nM (BRD2 BD1)，41 nM (BRD3 BD1)，41 nM (BRD4 BD1) 和143 nM (BRDT BD1)。

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GSK778 hydrochloride Chemical Structure

GSK778 hydrochloride Chemical Structure

CAS No. : 2863657-79-6

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GSK778 hydrochloride 的其他形式现货产品:

Other Forms of GSK778 hydrochloride:

GSK778 hydrochloride 相关抗体

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GSK778 (iBET-BD1) hydrochloride is a potent and selective BD1 bromodomain inhibitor of the BET proteins, with IC50s of 75 nM (BRD2 BD1), 41 nM (BRD3 BD1), 41 nM (BRD4 BD1), and 143 nM (BRDT BD1), respectively[1].

IC50 & Target

BRD2 BD1

75 nM (IC50)

BRD3 BD1

41 nM (IC50)

BRD4-BD1

41 nM (IC50)

BRDT BD1

143 nM (IC50)

分子量

548.08

Formula

C30H34ClN5O3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

GSK778 hydrochloride 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

GSK7782863657-79-6iBET-BD1GSK 778GSK-778ApoptosisEpigenetic Reader DomainBET-BD1Inhibitorinhibitorinhibit

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