2. Neuronal Signaling Immunology/Inflammation GPCR/G Protein
  3. Sigma Receptor Histamine Receptor
  4. KSK68

KSK68 是一种高亲和力双重 sigma-1 和 组胺 H3 受体拮抗剂，对 H3 受体、sigma-1、sigma-2 受体的 Ki 分别为 7.7 nM, 3.6 nM、22.4 nM。KSK68 对其他组胺受体亚型的亲和力可以忽略不计。KSK68 可用于伤害性疼痛和神经性疼痛的研究。

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KSK68 Chemical Structure

KSK68 Chemical Structure

CAS No. : 2566715-91-9

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KSK68 相关抗体

Top Publications Citing Use of Products

查看 Sigma Receptor 亚型特异性产品:

查看所有亚型
Sigma 1 Receptor Sigma 2 Receptor

查看 Histamine Receptor 亚型特异性产品:

查看所有亚型
H1 Receptor H2 Receptor H3 Receptor H4 Receptor Histamine Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

KSK68 is a high-affinity dual sigma-1 and histamine H3 receptor antagonist, with Kis of 7.7, 3.6, 22.4 nM for H3 receptor, sigma-1, sigma-2 receptor respectively. KSK68 has negligible affinity at the other histamine receptor subtypes. KSK68 can be used for research of nociceptive and neuropathic pain[1].

IC50 & Target

7.7 nM, 3.6 nM、22.4 nM (H3 receptor, sigma-1, sigma-2 receptor)[1]
分子量

364.48

Formula

C23H28N2O2
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

KSK68 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

KSK682566715-91-9KSK 68KSK-68Sigma ReceptorHistamine ReceptornociceptiveneuropathicpainhistamineInhibitorinhibitorinhibit

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HY-155614
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