2. GPCR/G Protein Neuronal Signaling
  3. mAChR
  4. Lu 26-046

Lu 26-046 是毒蕈碱型 M1 和 M2 受体 (M1 receptor，M2 receptor) 的激动剂，也是 M3 受体 (M3 receptor) 的弱拮抗剂，Ki 分别为 0.51、26 和 5 nM。Lu 26-046 表现出特异性刺激特性，可被大鼠识别。

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Lu 26-046 Chemical Structure

Lu 26-046 Chemical Structure

CAS No. : 143756-51-8

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Lu 26-046 相关抗体

Top Publications Citing Use of Products

查看 mAChR 亚型特异性产品:

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mAChR1 mAChR2 mAChR3 mAChR4 mAChR5

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Lu 26-046 is the agonist for muscarinic M1 receptor and M2 receptor and a weak antagonist for M3 receptor, with Ki of 0.51, 26 and 5 nM, respectively. Lu 26-046 exhibits specific stimulus property, that can be recognized by rats[1].

IC50 & Target

mAChR1

0.51 nM (Ki)

mAChR3

5 nM (Ki)

mAChR2

26 nM (Ki)

分子量

208.28

Formula

C10H12N2OS
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Lu 26-046 相关分类

  • 摩尔计算器

  • 稀释计算器

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Lu 26-046143756-51-8mAChRMuscarinic acetylcholine receptorguinea-pigWistar ratInhibitorinhibitorinhibit

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产品名称：
Lu 26-046
目录号：
HY-120329
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