2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. Masupirdine free base

Masupirdine free base  (Synonyms: SUVN-502 free base)

目录号: HY-109118
产品使用指南

摩尔计算器

Masupirdine free base (SUVN-502 free base) 是一种有效的，选择性的，具有口服生物可利用且可穿透脑屏障的5-HT6 受体拮抗剂 (对人 5-HT6 受体的 Ki 为 2.04 nM)。Masupirdine free base (SUVN-502 free base) 对 5-HT2A 受体和其他 100个 靶点显示高选择性，有研究阿尔茨海默病的潜力。

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Masupirdine free base Chemical Structure

Masupirdine free base Chemical Structure

CAS No. : 701205-60-9

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Masupirdine free base 的其他形式现货产品:

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Masupirdine free base 相关抗体

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5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Masupirdine free base (SUVN-502 free base) is a potent, selective, orally bioavailable, and brain penetrant 5-HT6 receptor antagonist (Ki of 2.04 nM for human 5-HT6 receptor). Masupirdine free base (SUVN-502 free base) shows high selectivity over 5-HT2A receptor and other 100 target sites, and has potential for treatment of Alzheimer's disease[1].

IC50 & Target[1]

5-HT6 Receptor

2.04 nM (Ki)

Clinical Trial
分子量

478.40

Formula

C21H24BrN3O3S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Masupirdine free base 相关分类

  • 摩尔计算器

  • 稀释计算器

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Masupirdine701205-60-9SUVN-502SUVN502SUVN 5025-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptorInhibitorinhibitorinhibit

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