2. GPCR/G Protein Neuronal Signaling
  3. Opioid Receptor
  4. MCOPPB

MCOPPB 是一种有口服活性的 Nociceptin/Orphanin FQ–Receptor 选择性激动剂。MCOPPB 通过小鼠大脑中的 NOP 受体抑制信号传导。MCOPPB 用于焦虑症研究。

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MCOPPB Chemical Structure

MCOPPB Chemical Structure

CAS No. : 1028969-49-4

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规格 是否有货
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MCOPPB 的其他形式现货产品:

Customer Review

Other Forms of MCOPPB:

MCOPPB 相关抗体

Top Publications Citing Use of Products

查看 Opioid Receptor 亚型特异性产品:

查看所有亚型
μ Opioid Receptor/MOR κ Opioid Receptor/KOR δ Opioid Receptor/DOR NOP Receptor/ORL1

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

MCOPPB is an orally active and selective agonist of Nociceptin/Orphanin FQ–Receptor. MCOPPB inhibits signaling through the NOP receptor in the mouse brain. MCOPPB is used in anxiety disorders research[1].

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
CHO-K1 EC50
34 nM
Compound: 1, MCOPPB
Agonist activity at human mu opioid receptor expressed in CHOK1 cells by [35S]GTPgammaS binding
Agonist activity at human mu opioid receptor expressed in CHOK1 cells by [35S]GTPgammaS binding
[PMID: 19125610]
CHO-K1 EC50
4696 nM
Compound: 1, MCOPPB
Agonist activity at human delta opioid receptor expressed in CHOK1 cells by [35S]GTPgammaS binding
Agonist activity at human delta opioid receptor expressed in CHOK1 cells by [35S]GTPgammaS binding
[PMID: 19125610]
HEK293 EC50
0.39 nM
Compound: 1, MCOPPB
Agonist activity at human NOP receptor expressed in HEK293 cells by [35S]GTPgammaS binding
Agonist activity at human NOP receptor expressed in HEK293 cells by [35S]GTPgammaS binding
[PMID: 19125610]
HEK293 EC50
80 nM
Compound: 1, MCOPPB
Agonist activity at human kappa opioid receptor expressed in HEK293 cells by [35S]GTPgammaS binding
Agonist activity at human kappa opioid receptor expressed in HEK293 cells by [35S]GTPgammaS binding
[PMID: 19125610]
分子量

408.62

Formula

C26H40N4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

MCOPPB 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

MCOPPB1028969-49-4Opioid ReceptorNociceptin/orphanin FQ peptide (NOP) receptorVogel conflict testAnxietyInhibitorinhibitorinhibit

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产品名称：
MCOPPB
目录号：
HY-10886
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