2. Metabolic Enzyme/Protease
  3. Phosphodiesterase (PDE)
  4. PDM-042

PDM-042 是一种有效的、选择性的、具有口服活性的磷酸二酯酶 10A (PDE10A) 抑制剂。PDM-042 对人和大鼠 PDE10A 显示出有效的抑制活性，IC50 值小于 1 nM，对其他磷酸二酯酶的选择性超过 1000 倍。 PDM-042可用于精神分裂症的研究。

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PDM-042 Chemical Structure

PDM-042 Chemical Structure

CAS No. : 1404488-48-7

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PDM-042 相关抗体

Top Publications Citing Use of Products

查看 Phosphodiesterase (PDE) 亚型特异性产品:

查看所有亚型
PDE1 PDE2 PDE3 PDE4 PDE5 PDE6 PDE7 PDE9 PDE10 PDE11 PDE12 PDE8 Autotaxin

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PDM-042 is a potent, selective, and orally active phosphodiesterase 10A (PDE10A) inhibitor. PDM-042 shows potent inhibitory activities for human and rat PDE10A with IC50 values of less than 1 nM and more than 1000-fold selectivity against other phosphodiesterases. PDM-042 can be used for the research of schizophrenia[1].

IC50 & Target

IC50: ＜1 nM (for human and rat PDE10A)[1]
分子量

406.48

Formula

C21H26N8O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

PDM-042 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PDM-0421404488-48-7PDM042PDM 042Phosphodiesterase (PDE)phosphodiesterase 10A (PDE10A)schizophreniaantipsychoticsPDM‐04Inhibitorinhibitorinhibit

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产品名称：
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目录号：
HY-160111
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