1. GPCR/G Protein Neuronal Signaling
  2. Opioid Receptor
  3. R-84760

R-84760 是一种选择性 κ-阿片受体 (κ-opioid receptor) 激动剂。R-84760 具有镇痛作用。

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R-84760 Chemical Structure

R-84760 Chemical Structure

CAS No. : 157824-23-2

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

R-84760 is a selective κ-opioid receptor agonist. R-84760 has antinociceptive effect[1][2].

IC50 & Target

κ Opioid Receptor/KOR

 

体外研究
(In Vitro)

在豚鼠脑膜部分的阿片受体结合试验中,R-84760 对 κ-阿片受体的亲和力比 CI-977 (HY-105235) 高 5 倍,R-84760 对 κ-阿片受体的选择性高于 U-69593 (HY-12363)[1]

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

435.84

Formula

C19H25Cl3N2OS

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Inquiry Information

产品名称:
R-84760
目录号:
HY-19206
需求量: