2. Metabolic Enzyme/Protease
  3. 11β-HSD
  4. (Rac)-BMS-816336

(Rac)-BMS-816336 (Compound 6n) 是 BMS-816336 的外消旋体。(Rac)-BMS-816336 是一种有效的人和小鼠 11β-羟类固醇脱氢酶 1 型 (11β-HSD1) 抑制剂，其 IC50 分别为 10 nM 和 68 nM，并具有良好的代谢稳定性 。

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(Rac)-BMS-816336 Chemical Structure

(Rac)-BMS-816336 Chemical Structure

CAS No. : 1009365-98-3

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规格 价格 是否有货
1 mg ￥1590
询问价格 & 货期
5 mg ￥3500
询问价格 & 货期
10 mg ￥5500
询问价格 & 货期

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Customer Review

Other Forms of (Rac)-BMS-816336:

(Rac)-BMS-816336 相关抗体

Top Publications Citing Use of Products

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

(Rac)-BMS-816336 (Compound 6n) is a racemate of BMS-816336. (Rac)-BMS-816336 is a potent inhibitor of human and mouse 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1) enzyme with IC50s of 10 nM and 68 nM, respectively. (Rac)-BMS-816336 has good metabolic stability[1].

IC50 & Target

IC50: 10 nM (Human 11β-HSD1) and 68 nM (Mouse 11β-HSD1)[1]
体内研究
(In Vivo)

(Rac)-BMS-816336 (compound 6n) has good metabolic stability, and the remaining rates in human, mouse and rats of 88%,82% and 72%, respectively[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

341.44

Formula

C21H27NO3
CAS 号
性状

固体

颜色

White to off-white

运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
纯度 & 产品资料
参考文献

(Rac)-BMS-816336 相关分类

  • 摩尔计算器

  • 稀释计算器

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

(Rac)-BMS-8163361009365-98-311β-HSD11beta-HSD11β-hydroxysteroid dehydrogenases11 beta-hydroxysteroid dehydrogenase11β-HSD1BMS-816336racematemetabolicstabilityInhibitorinhibitorinhibit

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产品名称：
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目录号：
HY-101930A
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