1. GPCR/G Protein Neuronal Signaling MAPK/ERK Pathway Stem Cell/Wnt
  2. Melanocortin Receptor ERK
  3. Resomelagon methanesulfonate

Resomelagon methanesulfonate  (Synonyms: AP1189 methanesulfonate)

目录号: HY-147301B
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Resomelagon methanesulfonate (AP1189 methanesulfonate) 是 Resomelagon (HY-147301) 的甲磺酸盐形式。Resomelagon methanesulfonate 是口服有效的黑皮质素受体 (MR) 激动剂。Resomelagon methanesulfonate 可诱导 ERK1/2 磷酸化和 Ca2+ 动员。Resomelagon methanesulfonate 在小鼠腹膜炎和关节炎模型中表现出抗炎活性。Resomelagon methanesulfonate 可用于肥胖和慢性炎症研究。

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Resomelagon methanesulfonate Chemical Structure

Resomelagon methanesulfonate Chemical Structure

CAS No. : 2933183-20-9

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Resomelagon methanesulfonate 的其他形式现货产品:

Other Forms of Resomelagon methanesulfonate:

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  • 生物活性

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  • 参考文献

生物活性

Resomelagon methanesulfonate (AP1189 methanesulfonate) is the methanesulfonate salt form of Resomelagon (HY-147301). Resomelagon methanesulfonate is an orally active melanocortin receptor (MR) agonist. Resomelagon methanesulfonate induces ERK1/2 phosphorylation and Ca2+ mobilization. Resomelagon methanesulfonate exhibits anti-inflammatory activity in mouse peritonitis and peritonitis model. Resomelagon methanesulfonate can be used for obesity and chronic inflammation research[1][2].

分子量

394.41

Formula

C15H18N6O5S

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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  • 稀释计算器

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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Resomelagon methanesulfonate
目录号:
HY-147301B
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