2. GPCR/G Protein Neuronal Signaling Anti-infection
  3. 5-HT Receptor Bacterial
  4. Trimipramine maleate (Standard)

Trimipramine maleate (Standard)  (Synonyms: 三甲丙咪嗪马来酸盐 (Standard))

目录号: HY-B1213R 纯度: ≥98%
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Trimipramine (maleate) (Standard) 是 Trimipramine (maleate) 的分析标准品。本产品用于研究及分析应用。Trimipramine maleate 是 5-HT 受体的拮抗剂，其对 5-HT1C，5-HT2 和 5-HT1A 受体的 pKi 值分别为 6.39，8.10，4.66。Trimipramine maleate 也是一种靶向人去甲肾上腺素 (hNAT)、血清素 (hSERT) 和有机阳离子转运体 (hOCT1、hOCT2) 的有选择性和强效的抑制剂，其 IC50 值分别为 4.99 μM、2.11 μM、3.72 μM、8.00 μM。Trimipramine maleate 具有血管活性和抗焦虑作用。

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Trimipramine maleate (Standard) Chemical Structure

Trimipramine maleate (Standard) Chemical Structure

CAS No. : 521-78-8

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生物活性

Trimipramine (maleate) (Standard) is the analytical standard of Trimipramine (maleate). This product is intended for research and analytical applications. Trimipramine maleate is a 5-HT receptor antagonist, with pKi binding values of 6.39, 8.10, 4.66 for 5-HT1C, 5-HT2 and 5-HT1A, respectively. Trimipramine maleate is also a potent and selective inhibitor targeting human noradrenaline (hNAT), serotonin (hSERT) and organic cation transporters (hOCT1, hOCT2) with IC50 values of 4.99 μM, 2.11 μM, 3.72 μM, 8.00 μM, respectively. Trimipramine maleate has vascular activity and anxiolytic efficacy.

分子量

410.51

Formula

C24H30N2O4
CAS 号
中文名称

马来酸三甲丙咪嗪 (Standard)；马来酸曲米帕明 (Standard)；三甲丙咪嗪马来酸盐 (Standard)
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
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Keywords:

Trimipramine maleate (Standard)521-78-8马来酸三甲丙咪嗪 (Standard)马来酸曲米帕明 (Standard)三甲丙咪嗪马来酸盐 (Standard)5-HT ReceptorBacterialSerotonin Receptor5-hydroxytryptamine Receptorantidepressants5-HT5-hydroxytryptamineserotonin5-HTlc receptors5-HTIA receptorsdopamineDADA D2 receptor5-HT1C5-HT25-HT1Aanxiolyticneurological diseasenoradrenalinehNAThSERThDAThuman organic cation transportershOCT1hOCT2hOCT3Inhibitorinhibitorinhibit

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