2. Membrane Transporter/Ion Channel Neuronal Signaling
  3. TRP Channel
  4. TRPC antagonist 1

TRPC antagonist 1 (compound 15g) 是一种有效的 TRP 通道 (TRPC) 拮抗剂，对 TRPC3、TRPC4、TRPC5、TPRC6 和 TRPC7 的 IC50 值分别为 2.4 μM、12.2 μM、7.6 μM、2.9 μM 和 3.4 μM。TRPC antagonist 1 在体外针对 U87 细胞系表现出显着的抗胶质母细胞瘤功效。

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TRPC antagonist 1 Chemical Structure

TRPC antagonist 1 Chemical Structure

CAS No. : 3027139-12-1

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TRPC antagonist 1 相关抗体

Top Publications Citing Use of Products

查看 TRP Channel 亚型特异性产品:

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TRPC TRPM TRPV TRPA TRPML

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

TRPC antagonist 1 (compound 15g) is a potent TRP channel (TRPC) antagonist with IC50s of 2.4 μM, 12.2 μM, 7.6 μM, 2.9 μM, and 3.4 μM for TRPC3, TRPC4, TRPC5, TPRC6, and TRPC7, respectively. TRPC antagonist 1 displays noteworthy anti-glioblastoma efficacy in vitro against U87 cell lines[1].

IC50 & Target[1]

TRPC3

2.4 μM (IC50)

TRPC4

12.2 μM (IC50)

TRPC5

7.6 μM (IC50)

TRPC6

2.9 μM (IC50)

TRPC7

3.4 μM (IC50)

分子量

418.51

Formula

C23H22N4O2S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

TRPC antagonist 1 相关分类

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  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

TRPC antagonist 13027139-12-1TRPC antagonist1TRPC antagonist-1TRP ChannelTransient receptor potential channelsTRPC antagonistanti-glioblastoma agentTRPC3TRPC4TRPC5TPRC6and TRPC7Inhibitorinhibitorinhibit

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TRPC antagonist 1
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