2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. WAY-100289

WAY-100289 是一种口服的 5-HT3 受体 (5-HT3 receptor) 拮抗剂，对分离的大鼠迷走神经具有高亲和力，pA2 为 8.9。WAY-100289 可抑制麻醉和清醒大鼠的 Bezold-Jarisch 反射。

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WAY-100289 Chemical Structure

WAY-100289 Chemical Structure

CAS No. : 136013-69-9

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WAY-100289 相关抗体

Top Publications Citing Use of Products

查看 5-HT Receptor 亚型特异性产品:

查看所有亚型
5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

WAY-100289 is an orally active antagonist for 5-HT3 receptor, that exhibits high affinity to the isolated rat vagus nerves with pA2 of 8.9. WAY-100289 inhibits the Bezold-Jarisch reflex in anesthetized and awake rats[1].

IC50 & Target

5-HT3 Receptor

 

分子量

357.45

Formula

C20H27N3O3
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

WAY-100289 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

WAY-100289136013-69-9WAY100289WAY 1002895-HT ReceptorSerotonin Receptor5-hydroxytryptamine Receptormigraineanxietymemory disordersvagus nerveorally activeInhibitorinhibitorinhibit

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产品名称：
WAY-100289
目录号：
HY-19136
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