2. GPCR/G Protein
  3. Adenosine Receptor
  4. Xanthine amine congener dihydrochloride

Xanthine amine congener dihydrochloride  (Synonyms: XAC dihydrochloride)

目录号: HY-110303
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Xanthine amine congener dihydrochloride (XAC dihydrochloride) 是一种有效的腺苷 A1 受体 (A1 receptor) 和 A2 受体 (A2 receptor) 拮抗剂，IC50 值分别为 1.8 和 114 nM。Xanthine amine congener 在动物实验模型中可作为惊厥剂。

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Xanthine amine congener dihydrochloride Chemical Structure

Xanthine amine congener dihydrochloride Chemical Structure

CAS No. : 1962928-23-9

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Xanthine amine congener dihydrochloride 的其他形式现货产品:

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Xanthine amine congener dihydrochloride 相关抗体

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生物活性

Xanthine amine congener dihydrochloride (XAC dihydrochloride) is a potent Adenosine A1 receptor and A2 receptor antagonist with IC50 values of 1.8 and 114 nM, respectively. Xanthine amine congener acts as a convulsant agent in mice model[1].

IC50 & Target

IC50: 1.8 nM (Adenosine A1 receptor)
IC50: 114 nM (Adenosine A2 receptor)[1]
体内研究
(In Vivo)

Xanthine amine congener dihydrochloride is more potent as a convulsant than either caffeine or theophyllin in infusion studies at the dosage 39.8 mg/kg. XAC has no effects by administering the drug via an i.p. injection, the seizure threshold >1000 mg/kg[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Mice[1]
Dosage: 39.8 mg/kg
Administration: Infusion injection; single dose
Result: Acted as a convulsant agent than either caffeine or theophyllin.
分子量

501.41

Formula

C21H30Cl2N6O4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Xanthine amine congener dihydrochloride 相关分类

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Xanthine amine congener1962928-23-9XACAdenosine ReceptorP1 receptorconvulsantAdenosine receptorantagonistInhibitorinhibitorinhibit

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