2. Metabolic Enzyme/Protease Neuronal Signaling
  3. Monoamine Oxidase Cytochrome P450
  4. 8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate

8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate 

目录号: HY-134664
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摩尔计算器

8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate 是一种不可逆的 CYP2A6?抑制剂，预孵育和共孵育的 IC50 分别为 8.64 μM 和 22.3 μM。8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate 也抑制 MAO-A 和 MAO-B，IC50 分别为 60.2 和 38.6 μM。

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8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate Chemical Structure

8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate Chemical Structure

CAS No. : 67667-71-4

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8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate 相关抗体

Top Publications Citing Use of Products

查看 Monoamine Oxidase 亚型特异性产品:

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MAO-A MAO-B

查看 Cytochrome P450 亚型特异性产品:

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CYP1 CYP2 CYP3 CYP4 CYP11 CYP17 Aromatase/CYP19A1 CYP26 CYP51 CYP2D6 CYP2C9 CYP2C19 CYP3A4 CYP17A1

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate is an irreversible CYP2A6 inhibitor with IC50s of 8.64 μM and 22.3 μM with pre-incubation and co-incubaition, respectively. 8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate also inhibits MAO-A and MAO-B with IC50s of 60.2 and 38.6 μM, respectively[1].

IC50 & Target

IC50: 8.64 μM (CYP2A6, pre-incubation), 22.3 μM (CYP2A6, co-incubation), 38.6 μM (MAO-B), 60.2 μM(MAO-A)[1]
Ki: 15.1 μM (CYP2A6), 27.2 μM (MAO-B), 60.2 μM (MAO-A)[1]
分子量

406.43

Formula

C21H26O8
CAS 号
结构分类
初始来源
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate 相关分类

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Keywords:

8α-(2-Methylacryloyloxy)-hirsutinolide-13-O-acetate67667-71-4Monoamine OxidaseCytochrome P450MAOCYPsP4502A6CYP2A6Vernonia cinereaasthmabronchitisInhibitorinhibitorinhibit

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