2. GPCR/G Protein Neuronal Signaling
  3. Adrenergic Receptor
  4. Dapiprazole

Dapiprazole  (Synonyms: 哌吡三唑；达哌唑)

目录号: HY-A0142
产品使用指南

摩尔计算器

Dapiprazole 是一种有效的、选择性的、具有口服活性的 α -1 肾上腺素受体 (alpha-1 adrenoceptor) 拮抗剂。Dapiprazole 抑制阿片类戒断症状。Dapiprazole 也可用作逆转瞳孔扩大的滴眼液。

在相同的摩尔浓度下，化合物盐形式与游离形式有相同的生物活性，但盐形式 Dapiprazole hydrochloride 通常具有更好的水溶性和稳定性。

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Dapiprazole Chemical Structure

Dapiprazole Chemical Structure

CAS No. : 72822-12-9

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Dapiprazole 的其他形式现货产品:

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Other Forms of Dapiprazole:

Dapiprazole 相关抗体

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α adrenergic receptor β adrenergic receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Dapiprazole is a potent, selective and orally active alpha-1 adrenoceptor antagonist. Dapiprazole suppresses the opioid withdrawal symptoms. Dapiprazole is also used as eye drops for reversing mydriasis[1][2][3].

IC50 & Target

α1-adrenergic receptor

 

体内研究
(In Vivo)

Dapiprazole hydrochloride (0-10 mg/kg or 0-3 mg/mice; i.p. or i.c.v.; once) reduces the overall severity of the opiate withdrawal symptoms in mice[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Swiss Albino male CD-1 mice weighing 20 -25 g, acute dependence model[1]
Dosage: 5, 7.5 and 10 mg/kg (i.p.) or 0.5, 1 and 3 mg/mice (i.c.v.), once
Administration: Intraperitoneal injection or intracerebroventricular administration, once
Result: Decreased jumping behavior, head shakes and paw shakes when administered just before naloxone.
分子量

325.45

Formula

C19H27N5
CAS 号
中文名称

哌吡三唑；达哌唑
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Dapiprazole 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Dapiprazole72822-12-9哌吡三唑达哌唑Adrenergic ReceptorBeta Receptoropioid withdrawalmydriasisInhibitorinhibitorinhibit

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