2. GPCR/G Protein Metabolic Enzyme/Protease MAPK/ERK Pathway
  3. Phosphodiesterase (PDE) Ras
  4. Deltarasin trihydrochloride

Deltarasin 是一种 KRAS-PDEδ 相互作用的抑制剂，能够与 PDEδ 结合，Kd 值为 38 nM。Deltarasin 可用于癌症的研究。

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Deltarasin trihydrochloride Chemical Structure

Deltarasin trihydrochloride Chemical Structure

CAS No. : 1440898-82-7

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Deltarasin trihydrochloride 的其他形式现货产品:

Other Forms of Deltarasin trihydrochloride:

Deltarasin trihydrochloride 相关抗体

Top Publications Citing Use of Products

MCE 顾客使用本产品发表的 2 篇科研文献

查看 Phosphodiesterase (PDE) 亚型特异性产品:

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PDE1 PDE2 PDE3 PDE4 PDE5 PDE6 PDE7 PDE9 PDE10 PDE11 PDE12 PDE8 Autotaxin

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K-Ras H-Ras N-Ras Ras

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Deltarasin is an inhibitor of KRAS-PDEδ interaction with Kd of 38 nM for binding to purified PDEδ. Deltarasin can be used in the study of cancer.

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
A549 IC50
6.4 μM
Compound: Deltarasin
Antiproliferative activity against human A549 cells harboring KRAS G12S point mutant after 72 hrs by SRB assay
Antiproliferative activity against human A549 cells harboring KRAS G12S point mutant after 72 hrs by SRB assay
[PMID: 30562696]
分子量

713.14

Formula

C40H40Cl3N5O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Deltarasin trihydrochloride 相关分类

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  • Do most proteins show cross-species activity?

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Keywords:

Deltarasin trihydrochloride1440898-82-7Phosphodiesterase (PDE)RascancerInhibitorinhibitorinhibit

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