1. Epigenetics
  2. Histone Methyltransferase
  3. EPZ028862

EPZ028862 是一种选择性的 SMYD3 抑制剂,可用于癌症研究。

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EPZ028862 Chemical Structure

EPZ028862 Chemical Structure

CAS No. : 1887082-53-2

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规格 是否有货
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Customer Review

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

EPZ028862 is a selective SMYD3 inhibitor for cancer research[1].

体内研究
(In Vivo)

The pharmacokinetic parameters of EPZ028862( IV: 1 mg/kg; PO: 5 mg/kg)

Parameter Mouse Rat Dog Cynomolgus
CLp(mL/min/kg) 79.8 32.7 13.9 21.4
CLr(mL/min/kg) 23.6 21 1.97 1.06
Vss(L/kg) 9.5 4.4 5.8 9.5
t1/2(h) 2 2.1 5.4 5.6
MRT(h) 2 59 7 7.4
tmax(h) 0.33 1 1.5 2
F(%) 100 59 70 62

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

分子量

422.54

Formula

C20H30N4O4S

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
EPZ028862
目录号:
HY-145444
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