2. GPCR/G Protein Neuronal Signaling
  3. Cholecystokinin Receptor
  4. Gastrazole

Gastrazole  (Synonyms: JB95008)

目录号: HY-19445
产品使用指南

摩尔计算器

Gastrazole (JB95008) 是一种有效的和选择性的 CCK2/gastrin 受体拮抗剂。Gastrazole 可降低胃酸水平。Gastrazole 抑制胃泌素刺激的胰腺癌生长。

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Gastrazole Chemical Structure

Gastrazole Chemical Structure

CAS No. : 862583-15-1

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Other Forms of Gastrazole:

Gastrazole 相关抗体

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CCKAR CCKBR

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

Gastrazole (JB95008) is potent and selective CCK2/gastrin receptor antagonist. Gastrazole can decrease the level of gastric acid. Gastrazole inhibits the Gastrin-stimulated growth of pancreatic cancer[1][2].

IC50 & Target

CCK2/gastrin receptor[1]
体内研究
(In Vivo)

Gastrazole (0.15-3 μmol/kg; i.v.) dose-dependently inhibits the Pentagastrin-stimulated gastric acid secretion[2].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male Sprague-Dawley rats with a gastric fistula[2]
Dosage: 0.15, 0.3, 3 mg/kg
Administration: Intravenous administration
Result: Dose-dependently inhibited Pentagastrin-stimulation acid secretion by maximally 73%.
分子量

687.63

Formula

C34H32FN5Na2O7
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

Gastrazole 相关分类

  • 摩尔计算器

  • 稀释计算器

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Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Gastrazole862583-15-1JB95008JB 95008JB-95008Cholecystokinin ReceptorCCK ReceptorCCK2gastrinpancreaticcancerInhibitorinhibitorinhibit

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