1. GPCR/G Protein Immunology/Inflammation Neuronal Signaling Membrane Transporter/Ion Channel
  2. mAChR CRAC Channel Histamine Receptor
  3. GS 283

GS 283 是一种具有钙拮抗作用以及弱组胺和毒蕈碱受体阻断活性的化合物,具有调节豚鼠和大鼠气管平滑肌收缩的活性。GS 283可抑制豚鼠和大鼠气管平滑肌中由卡巴胆碱、组胺(仅豚鼠)和高K?诱导的收缩,在豚鼠气管平滑肌中可抑制Ca2?诱导的收缩,高浓度时可完全消除卡巴胆碱在无Ca2?介质中诱导的收缩。

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GS 283 Chemical Structure

GS 283 Chemical Structure

CAS No. : 149440-36-8

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  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

GS 283 is a compound with calcium antagonist and weak histamine and muscarinic receptor blocking activity, with activity in modulating contraction of guinea pig and rat tracheal smooth muscle. GS 283 inhibits contractions induced by carbachol, histamine (guinea pig only), and high K? in guinea pig and rat tracheal smooth muscle, inhibits Ca2?-induced contractions in guinea pig tracheal smooth muscle, and at high concentrations completely abolishes contractions induced by carbachol in Ca2?-free medium.

分子量

313.30

Formula

C17H15NO5

CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.

储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.

纯度 & 产品资料
参考文献
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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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产品名称:
GS 283
目录号:
HY-114743
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