2. GPCR/G Protein
  3. Adenosine Receptor
  4. LAS38096

LAS38096 是有效的、选择性的 A2B 腺苷受体的拮抗剂，其 Ki 值为 17 nM。

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LAS38096 Chemical Structure

LAS38096 Chemical Structure

CAS No. : 851371-22-7

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规格 价格 是否有货 数量
1 mg ￥3995
1 - 2 周
5 mg   询价  
10 mg   询价  

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Customer Review

LAS38096 相关抗体

Top Publications Citing Use of Products

查看 Adenosine Receptor 亚型特异性产品:

查看所有亚型
Adenosine A1 receptor (A1R) Adenosine A2A receptor (A2AR) Adenosine A2B receptor (A2BR) Adenosine A3 receptor (A3R)

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

LAS38096 is a potent, selective, and efficacious A2B Adenosine Receptor antagonist, with a Ki of 17 nM[1].
IC50 & Target[1].

A2B

17 nM (Ki)

A1

>1000 nM (Ki)

A2A

>2500 nM (Ki)

A3

>1000 nM (Ki)

细胞效力
(Cellular Effect)
Cell Line Type Value Description References
CHO IC50
349 nM
Compound: 5, LAS38096
Activity at mouse A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
Activity at mouse A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
[PMID: 17469811]
HEK293 IC50
321 nM
Compound: 5, LAS38096
Activity at human A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
Activity at human A2B receptor expressed in HEK293 cells assessed as inhibition of NECA-induced intracellular cAMP levels by ELISA
[PMID: 17469811]
分子量

316.32

Formula

C17H12N6O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

LAS38096 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

LAS38096851371-22-7LAS 38096LAS-38096Adenosine ReceptorP1 receptorA2BInhibitorinhibitorinhibit

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产品名称：
LAS38096
目录号：
HY-111295
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