2. GPCR/G Protein Neuronal Signaling
  3. 5-HT Receptor
  4. LY302148

LY302148 是 5-HT1F 的受体配体。与 5-HT 的 Emax 相比，LY302148 表现为 5-HT1F 受体的部分激动剂。在针对人 5-HT1F 受体的 [35S]GTPγS 结合试验中，LY302148 表现出较好的效力，其 EC50 值为 5.23 nM。LY302148 可以用于偏头痛的研究。

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LY302148 Chemical Structure

LY302148 Chemical Structure

CAS No. : 182564-47-2

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LY302148 相关抗体

Top Publications Citing Use of Products

查看 5-HT Receptor 亚型特异性产品:

查看所有亚型
5-HT1 Receptor 5-HT2 Receptor 5-HT3 Receptor 5-HT4 Receptor 5-HT5 Receptor 5-HT6 Receptor 5-HT7 Receptor 5-HT Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

LY302148 is a receptor ligand for 5-HT1F. Compared to the Emax of 5-HT, LY302148 behaves as a partial agonist for the 5-HT1F receptor. In the [35S]GTPγS binding assay targeting human 5-HT1F receptors, LY302148 exhibits good potency with an EC50 value of 5.23 nM. LY302148 can be used in the research of migraine[1].

分子量

326.41

Formula

C19H23FN4
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

LY302148 相关分类

  • 摩尔计算器

  • 稀释计算器

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Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

LY302148182564-47-2LY 302148LY-3021485-HT ReceptorSerotonin Receptor5-hydroxytryptamine ReceptormigraineInhibitorinhibitorinhibit

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HY-114678
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