2. GPCR/G Protein Neuronal Signaling Immunology/Inflammation
  3. Histamine Receptor
  4. ROS 234

ROS 234 是有效的 H3 拮抗剂，对豚鼠回肠 H3 受体的pKB 值为 9.46，大鼠大脑的 pKi 值为 8.90，离体大鼠大脑皮层的 ED50 值为 19.12 mg/kg (腹腔注射)。ROS 234 具有较差的中枢通路。

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ROS 234 Chemical Structure

ROS 234 Chemical Structure

CAS No. : 184576-87-2

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Other Forms of ROS 234:

ROS 234 相关抗体

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H1 Receptor H2 Receptor H3 Receptor H4 Receptor Histamine Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

ROS 234 is a potent H3 antagonist, with a pKB of 9.46 for Guinea-pig ileum H3-receptor, a pKi of 8.90 for Rat cerebral cortex H3-receptor, and a ED50 of 19.12 mg/kg (ip) in ex vivo of Rat cerebral cortex. ROS 234 diaplays poor central access[1][2].

IC50 & Target[1]

rat H3 receptor

8.90 (pKi)

体内研究
(In Vivo)

ROS 234 centrally injected, significantly shortens pentobarbital narcosis[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

241.29

Formula

C13H15N5
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

ROS 234 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

ROS 234184576-87-2ROS234ROS-234Histamine Receptorguinea-pig ileumRat cerebral cortex HRat cerebral cortexcentral accessInhibitorinhibitorinhibit

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