2. GPCR/G Protein Neuronal Signaling
  3. Cholecystokinin Receptor
  4. TP-680

TP-680 是一种胆囊收缩素受体 (cholecystokinin receptor) 拮抗剂。TP-680 与大鼠胰腺 CCKA 受体 (IC50=1.2 nM) 的结合强度是与大鼠大脑 CCKB 受体 (IC50=1812.5 nM) 的结合强度的 1510 倍。TP-680 可用于胃肠道疾病的研究。

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TP-680 Chemical Structure

TP-680 Chemical Structure

CAS No. : 176915-07-4

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TP-680 相关抗体

Top Publications Citing Use of Products

查看 Cholecystokinin Receptor 亚型特异性产品:

查看所有亚型
CCKAR CCKBR

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

TP-680 is a cholecystokinin receptor antagonist. TP-680 binds 1510 times more strongly to rat pancreatic CCKA receptors (IC50=1.2 nM) than to rat brain CCKB receptors (IC50=1812.5 nM). TP-680 can be used in the study of gastrointestinal diseases[1].

IC50 & Target[1]

CCKAR

1.2 nM (IC50)

CCKBR

1812.5 nM (IC50)

分子量

619.73

Formula

C35H33N5O4S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

TP-680 相关分类

  • 摩尔计算器

  • 稀释计算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

质量   浓度   体积   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

浓度 (start) × 体积 (start) = 浓度 (final) × 体积 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

TP-680176915-07-4TP680TP 680Cholecystokinin ReceptorCCK ReceptorCholecystokininantagonistgastrointestinal diseasesCCKACCKBInhibitorinhibitorinhibit

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产品名称：
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目录号：
HY-119127
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