2. GPCR/G Protein
  3. P2Y Receptor
  4. PSB-1114 tetrasodium

PSB-1114 tetrasodium 是一种有效的，酶促稳定的亚型选择性 P2Y2 受体激动剂，EC50 为 134 nM。PSB-1114 tetrasodium 相对于 P2Y4 (EC50 为 9.3 μM) 和 P2Y6 (EC50 为 7.0 μM) 受体显示出 50 倍以上的选择性。

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PSB-1114 tetrasodium Chemical Structure

PSB-1114 tetrasodium Chemical Structure

CAS No. : 1657025-60-9

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PSB-1114 tetrasodium 的其他形式现货产品:

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PSB-1114 tetrasodium 相关抗体

Top Publications Citing Use of Products

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P2Y1 Receptor P2Y2 Receptor P2Y6 Receptor P2Y12 Receptor P2Y13 Receptor P2Y14 Receptor

  • 生物活性

  • 纯度 & 产品资料

  • 参考文献

生物活性

PSB-1114 tetrasodium is a potent, enzymatically stable, and subtype-selective P2Y2 receptor agonist with an EC50 of 134 nM. PSB-1114 tetrasodium displays >50-fold selectivity versus the P2Y4 (EC50 of 9.3 μM) and P2Y6 (EC50 of 7.0 μM) receptors[1].

IC50 & Target

EC50: 134 nM (P2Y2 receptor), 9.3 μM (P2Y4 receptor); 7.0 μM (P2Y6 receptor)[1]
体外研究
(In Vitro)

PSB-1114 (4-Thio-β,γ-difluoromethylene-UTP; compound 14g) displays >60-fold selectivity versus P2Y4 and P2Y6 receptors. Because of its high potency, selectivity, and expected metabolic stability toward ectonucleotidases, in particular NTPDases, PSB-1114 may be a useful pharmacological tool for studying P2Y2 receptors[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

PSB-1114 tetrasodium 相关抗体:
分子量

622.14

Formula

C10H11F2N2Na4O13P3S
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料
参考文献

PSB-1114 tetrasodium 相关分类

  • 摩尔计算器

  • 稀释计算器

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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PSB-1114 tetrasodium1657025-60-9P2Y ReceptorP2Y2commercialsourcesectonucleotidasestablemetabolicInhibitorinhibitorinhibit

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