1. Signaling Pathways
  2. GPCR/G Protein
  3. P2Y Receptor
  4. P2Y Receptor Inhibitors

P2Y Receptor Inhibitors

P2Y1 Receptor

P2Y2 Receptor

P2Y6 Receptor

P2Y12 Receptor

P2Y13 Receptor

P2Y14 Receptor

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

P2Y Receptor Inhibitors, Agonists, Antagonists, Activators & Modulators
Product Name P2Y1 Receptor P2Y2 Receptor P2Y6 Receptor P2Y12 Receptor P2Y13 Receptor P2Y14 Receptor Purity
Ticagrelor      
P2Y12 Receptor
    99.98%
Clopidogrel      
P2Y12 Receptor
    99.57%
Uridine 5′-diphosphoglucose disodium salt          
P2Y14 Receptor
99.82%
P2Y14R antagonist 1
P2Y1 Receptor, IC50: > 100 nM
P2Y2 Receptor, IC50: > 100 nM
P2Y6 Receptor, IC50: 89.7 nM
P2Y12 Receptor, IC50: > 100 nM
 
P2Y14 Receptor, IC50: 0.6 nM
MRS 2578    
P2Y6 Receptor
      98.15%
UDP-Galactose disodium          
P2Y14 Receptor, EC50: 0.67 μM
99.42%
Uridine-5'-diphosphate disodium salt    
P2Y6 Receptor
      ≥99.0%
YM-254890
P2Y1 Receptor
          ≥99.0%
Cangrelor tetrasodium      
P2Y12 Receptor
    99.93%
PPTN hydrochloride          
P2Y14 Receptor
99.89%
Clopidogrel hydrogen sulfate      
P2Y12 Receptor
    99.43%
Diquafosol tetrasodium  
P2Y2 Receptor
        ≥99.0%
PSB-0739      
P2Y12 Receptor
    98.67%
AR-C118925XX  
P2Y2 Receptor
        ≥99.0%
Prasugrel      
P2Y12 Receptor
    99.85%
2-Methylthio-AMP      
P2Y12 Receptor
    99.30%
Prasugrel hydrochloride      
P2Y12 Receptor
    98.90%
MRS2500 tetraammonium
P2Y1 Receptor
          99.85%
Clopidogrel thiolactone      
P2Y12 Receptor
    ≥98.0%
PIT
P2Y1 Receptor, IC50: 0.14 μM μM
          98.57%
2-MeS-ADP trisodium      
P2Y12 Receptor
P2Y13 Receptor
  98.70%
AZD1283      
P2Y12 Receptor, IC50: 11 nM
    99.27%
MRS2365
P2Y1 Receptor, EC50: 0.4 nM
         
MRS2365 trisodium
P2Y1 Receptor, EC50: 0.4 nM
          ≥99.0%
MRS2279 diammonium
P2Y1 Receptor, IC50: 51.6 nM
          ≥98.0%
MRS2768 tetrasodium salt  
P2Y2 Receptor
        98.70%
Prasugrel-d3      
P2Y12 Receptor
    98.58%
2-Methylthio-AMP diTEA      
P2Y12 Receptor
    ≥98.0%
Uridine diphosphate glucose          
P2Y14 Receptor
ADP-β-S trilithium      
P2Y12 Receptor
   
Adenosine 2',5'-diphosphate sodium
P2Y1 Receptor
          ≥99.0%
4-Thiouridine 5′-triphosphate tetralithium  
P2Y2 Receptor, EC50: 35 nM
       
Cangrelor      
P2Y12 Receptor
   
HDL-16          
P2Y14 Receptor, IC50: 0.3095 nM
P2Y14R antagonist 2          
P2Y14 Receptor, IC50: 0.40 nM
UDP-Galactose          
P2Y14 Receptor, EC50: 0.67 μM
Regrelor disodium      
P2Y12 Receptor
   
4-Thiouridine 5′-triphosphate tetrasodium  
P2Y2 Receptor, EC50: 35 nM
       
Prasugrel-d5      
P2Y12 Receptor
   
MRS-2179
P2Y1 Receptor
         
2-MeSADP      
P2Y12 Receptor, EC50: 5 nM
P2Y13 Receptor, EC50: 19 nM
 
Blue FPG-A trisodium
P2Y1 Receptor, IC50: 2.6 μM
         
MRS2693 ammonium    
P2Y6 Receptor, EC50: 0.015 μM
     
MRS2279
P2Y1 Receptor, IC50: 51.6 nM
         
5-OMe-UDP    
P2Y6 Receptor, EC50: 0.08 μM
     
Uridine 5′-diphosphoglucose-13C disodium    
P2Y6 Receptor
     
MRS2496
P2Y1 Receptor
         
Sp-UTP-α-S  
P2Y2 Receptor
       
Prasugrel (Maleic acid)      
P2Y12 Receptor
   
Diquafosol  
P2Y2 Receptor
       
MRS2603
P2Y1 Receptor
     
P2Y13 Receptor
 
Elinogrel potassium      
P2Y12 Receptor
   
Ticagrelor-d7      
P2Y12 Receptor
   
2-Thio-UTP  
P2Y2 Receptor, EC50: 50 nM