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  3. Others
  4. (R)-KT109

(R)-KT109 是一种高效二酰甘油脂肪酶 β (DAGLβ) 抑制剂，IC50 为 0.79 nM，可有效阻断 DAGLα 介导的 1-硬脂酰-2-花生四烯酰-sn-甘油水解。此外，它还表现出对 α/β-水解酶结构域蛋白 6 (ABHD6) 的抑制活性，IC50 为 2.51 nM，与 (S) 异构体 (S)-KT109 相比，对 DAGLβ、DAGLα 和 ABHD6 的效力更强。

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(R)-KT109 Chemical Structure

(R)-KT109 Chemical Structure

CAS No. : 2055172-60-4

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(R)-KT109 相关抗体

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  • 生物活性

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生物活性

(R)-KT109 is a highly potent inhibitor of diacylglycerol lipase β (DAGLβ) with an IC50 of 0.79 nM and effectively blocks DAGLα-mediated hydrolysis of 1-stearoyl-2-arachidonoyl-sn-glycerol. Additionally, it demonstrates inhibitory activity against α/β-hydrolase domain-containing protein 6 (ABHD6) with an IC50 of 2.51 nM, exhibiting greater potency for DAGLβ, DAGLα, and ABHD6 compared to its (S) isomer, (S)-KT109.

分子量

422.52

Formula

C27H26N4O
CAS 号
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
纯度 & 产品资料

(R)-KT109 相关分类

  • 摩尔计算器

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Keywords:

(R)-KT1092055172-60-4OthersInhibitorinhibitorinhibit

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